Fragment-Based Discovery of a Dual pan-RET/VEGFR2 Kinase Inhibitor Optimized for Single-Agent Polypharmacology

Brendan Frett, Francesca Carlomagno, Maria Luisa Moccia, Annalisa Brescia, Giorgia Federico, Valentina De Falco, Brittany Admire, Zhongzhu Chen, Wenqing Qi, Massimo Santoro, Hong Yu Li

Research output: Contribution to journalArticle

4 Scopus citations
Original languageEnglish (US)
JournalAngewandte Chemie - International Edition
DOIs
StateAccepted/In press - 2015

ASJC Scopus subject areas

  • Chemistry(all)
  • Catalysis

Cite this

Frett, B., Carlomagno, F., Moccia, M. L., Brescia, A., Federico, G., De Falco, V., Admire, B., Chen, Z., Qi, W., Santoro, M., & Li, H. Y. (Accepted/In press). Fragment-Based Discovery of a Dual pan-RET/VEGFR2 Kinase Inhibitor Optimized for Single-Agent Polypharmacology. Angewandte Chemie - International Edition. https://doi.org/10.1002/anie.201505540